SCHEMBL8624915

SCHEMBL8624915

CC(Nc1c(C(N)c2ccc(C#N)cc2Cl)c(=O)c1=O)C(C)(C)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 1/20 0.42
ABCC8 Q09428 1/20 0.42
KCNJ11 Q14654 1/20 0.42
KCNJ8 Q15842 1/20 0.42
PDK1 Q15118 1/20 0.38
PDK2 Q15119 1/20 0.38
PDK3 Q15120 1/20 0.38
PDK4 Q16654 1/20 0.38
HSD11B1 P28845 1/20 0.36
SLC22A12 Q96S37 2/20 0.34
TNF P01375 2/20 0.33
NR3C1 P04150 2/20 0.32
CYP2C9 P11712 1/20 0.32
KCNH2 Q12809 1/20 0.32
CNR2 P34972 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
MTOR P42345 1/20 0.32
PIK3CG P48736 1/20 0.32
PRKDC P78527 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619019 0.91 ABCC9 (0.51) ABCC9ABCC8KCNJ11KCNJ8PDK1
SCHEMBL4261010 0.79 ABCC9 (0.40) ABCC9ABCC8KCNJ11KCNJ8PDK1
SCHEMBL8622441 0.78 PDK1 (0.38) ABCC9ABCC8KCNJ11KCNJ8PDK1
SCHEMBL7894099 0.77 ABCC9 (0.50) ABCC9ABCC8KCNJ11KCNJ8PDK1
SCHEMBL8667527 0.72 ABCC9 (0.51) ABCC9ABCC8KCNJ11KCNJ8HSD11B1
SCHEMBL8624137 0.69 ABCC9 (0.41) ABCC9ABCC8KCNJ11KCNJ8SLC22A12
SCHEMBL8420167 0.69 ABCC9 (0.48) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL26916884 0.68 LMNA (0.58) PDK1PDK2PDK3PDK4HSD11B1
SCHEMBL26620605 0.68 LMNA (0.58) PDK1PDK2PDK3PDK4HSD11B1
SCHEMBL7895113 0.68 ABCC9 (0.60) ABCC9ABCC8KCNJ11KCNJ8PDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780505-A ADMINISTERING AS SMOOTH MUSCLE RELAXANT AMERICAN HOME PRODUCTS CORPORATION (US) 1998-07-14 US claimed