SCHEMBL8625475

SCHEMBL8625475

COc1ccc(S(=O)(=O)Nc2ccccc2NC(=O)c2cc(C)nc(Cl)c2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
HDAC3 O15379 3/20 0.52
HDAC1 Q13547 3/20 0.52
NCOR2 Q9Y618 3/20 0.52
HDAC2 Q92769 2/20 0.52
KEAP1 Q14145 1/20 0.51
GFER P55789 1/20 0.50
SMN1; SMN2 Q16637 3/20 0.49
F10 P00742 1/20 0.49
LMNA P02545 3/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
TP53 P04637 1/20 0.48
HPGD P15428 1/20 0.48
HTT P42858 1/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
TUBB4A P04350 1/20 0.47
TUBB P07437 1/20 0.47
TUBA3C P0DPH7 1/20 0.47
TUBA1B P68363 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30926697 0.82 F10 (0.64) ALDH1A1HDAC3HDAC1NCOR2HDAC2
SCHEMBL27180977 0.82 F10 (0.64) ALDH1A1HDAC3HDAC1NCOR2HDAC2
SCHEMBL8626468 0.82 SMN1; SMN2 (0.69) ALDH1A1HDAC3HDAC1NCOR2HDAC2
SCHEMBL8625192 0.81 F10 (0.67) ALDH1A1HDAC3HDAC1NCOR2HDAC2
SCHEMBL8625679 0.78 TUBB4A (0.68) ALDH1A1HDAC3HDAC1NCOR2HDAC2
SCHEMBL8625306 0.78 MEN1 (0.61) ALDH1A1HDAC3HDAC1NCOR2HDAC2
SCHEMBL8627623 0.77 F10 (0.64) ALDH1A1HDAC3HDAC1NCOR2HDAC2
SCHEMBL8626109 0.77 CCR9 (0.66) KEAP1SMN1; SMN2HPGDMEN1KMT2A
SCHEMBL6562129 0.77 LMNA (0.55) ALDH1A1HDAC3HDAC1NCOR2HDAC2
SCHEMBL8628089 0.77 MAPT (0.60) ALDH1A1HDAC3HDAC1NCOR2HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0472053-B1 Sulfonamide derivatives EISAI CO LTD (JP) 1998-06-17 EP disclosed
US-5610304-A Pyrimidinyl or pyridinyl sulfonamide substituted compounds EISAI CO., LTD. (JP) 1997-03-11 US disclosed
US-5610320-A ANTITUMOR AGENTS EISAI CO., LTD. (JP) 1997-03-11 US disclosed
US-5434172-A Antitumor EISAI CO., LTD. (JP) 1995-07-18 US disclosed
US-5332751-A Antitumor EISAI CO., LTD. (JP) 1994-07-26 US disclosed
US-5292758-A Sulfonamide derivatives EISAI CO., LTD. (JP) 1994-03-08 US disclosed
US-5250549-A Antitumor agents EISAI CO., LTD. (JP) 1993-10-05 US disclosed
EP-0472053-A2 Sulfonamide derivatives Eisai Co., Ltd. (JP) 1992-02-26 EP disclosed