SCHEMBL8625869

SCHEMBL8625869

Clc1ccc(-c2sccc2-c2nn[c]o2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 6/20 0.40
PTGS2 P35354 2/20 0.35
MAPK14 Q16539 1/20 0.35
RAB9A P51151 4/20 0.32
NPC1 O15118 3/20 0.32
TSHR P16473 3/20 0.32
HSD17B10 Q99714 3/20 0.32
KDM4E B2RXH2 3/20 0.32
TP53 P04637 2/20 0.32
ALDH1A1 P00352 2/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
SENP8 Q96LD8 1/20 0.32
SENP7 Q9BQF6 1/20 0.32
SENP6 Q9GZR1 1/20 0.32
NOTUM Q6P988 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PTGS1 P23219 4/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL344372 0.77 NPC1 (0.46) CASP3PTGS2RAB9ANPC1TSHR
SCHEMBL4552995 0.63 CASP3 (0.59) CASP3RAB9ANPC1TSHRHSD17B10
SCHEMBL8985534 0.63 PTGS1 (0.71) PTGS2MAPK14RAB9APTGS1
SCHEMBL15286968 0.62 NPC1 (0.54) RAB9ANPC1TSHRTP53NFKB1
SCHEMBL18005410 0.61 PTGS1 (0.39) CASP3PTGS2MAPK14KDM4EALDH1A1
SCHEMBL7457943 0.61 CASP3 (0.41) CASP3PTGS2RAB9ANPC1TSHR
SCHEMBL10407505 0.61 CYP2A6 (0.52) CASP3PTGS2
SCHEMBL3619389 0.60 RAB9A (0.44) CASP3RAB9ANPC1TSHRHSD17B10
SCHEMBL547061 0.60 CYP2A6 (0.50) CASP3PTGS2RAB9AALDH1A1SMN1; SMN2
SCHEMBL7223282 0.59 NPC1 (0.47) RAB9ANPC1TSHRHSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE35754-E FOR TREATING BACTERIAL INFECTIONS HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-24 US disclosed
US-5710146-A ANTIBIOTICS FOR BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1998-01-20 US disclosed
US-5089490-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1992-02-18 US disclosed
US-4758556-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1988-07-19 US disclosed
US-4399131-A Cephem derivatives HOECHST AG (DE) 1983-08-16 US disclosed
US-4278793-A ANTIBIOTICS, BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1981-07-14 US disclosed