SCHEMBL8627674

SCHEMBL8627674

Cc1ccc(S(=O)(=O)OCCCOC2CCc3cc(Cl)ccc3N(C(=O)c3ccc([N+](=O)[O-])cc3C)C2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 2/20 0.38
DRD4 P21917 1/20 0.35
ALDH1A1 P00352 6/20 0.34
LMNA P02545 4/20 0.34
RAB9A P51151 2/20 0.34
PAX8 Q06710 2/20 0.34
RECQL P46063 1/20 0.34
FLT1 P17948 1/20 0.33
FLT4 P35916 1/20 0.33
KDR P35968 1/20 0.33
TP53 P04637 2/20 0.33
GAA P10253 1/20 0.33
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
NFKB1 P19838 1/20 0.33
CYP2C19 P33261 1/20 0.33
HTT P42858 1/20 0.33
NFKB2 Q00653 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634460 0.92 MAPT (0.36) DRD4ALDH1A1TP53GAAMEN1
SCHEMBL8630394 0.91 ALDH1A1 (0.34) ALDH1A1LMNARAB9APAX8RECQL
SCHEMBL8629473 0.89 AVPR2 (0.51) AVPR2LMNATP53ESR1ESR2
SCHEMBL8627677 0.86 AVPR2 (0.38) AVPR2DRD4ALDH1A1LMNARAB9A
SCHEMBL8627671 0.85 AVPR2 (0.37) AVPR2DRD4ALDH1A1LMNARAB9A
SCHEMBL4681642 0.82 AVPR2 (0.41) AVPR2ALDH1A1LMNARAB9APAX8
SCHEMBL8634051 0.82 AVPR2 (0.42) AVPR2TP53SMN1; SMN2MAPT
SCHEMBL8627401 0.81 AVPR2 (0.39) AVPR2DRD4ALDH1A1LMNARAB9A
SCHEMBL8630680 0.79 AVPR2 (0.38) AVPR2ALDH1A1LMNARAB9APAX8
SCHEMBL8634457 0.79 TP53 (0.34) AVPR2DRD4ALDH1A1TP53GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed