SCHEMBL8634457

SCHEMBL8634457

CCC(OC1CCc2cc(Cl)ccc2N(C(=O)c2ccc([N+](=O)[O-])cc2OC)C1)OS(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.34
MAPT P10636 2/20 0.34
KCNMA1 Q12791 1/20 0.34
ALDH1A1 P00352 3/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
IDH1 O75874 1/20 0.33
PYGL P06737 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP3A4 P08684 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
DRD4 P21917 1/20 0.33
AVPR2 P30518 1/20 0.33
SCN5A Q14524 1/20 0.32
SCN9A Q15858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8627671 0.93 AVPR2 (0.37) TP53MAPTALDH1A1GAAMEN1
SCHEMBL8634049 0.90 AVPR2 (0.42) TP53MAPTGAAAVPR2SCN5A
SCHEMBL8634460 0.85 MAPT (0.36) TP53MAPTKCNMA1ALDH1A1POLB
SCHEMBL8630392 0.85 ALDH1A1 (0.34) TP53MAPTALDH1A1GAAMEN1
SCHEMBL8629470 0.84 AVPR2 (0.50) TP53MAPTAVPR2SCN5ASCN9A
SCHEMBL8627674 0.79 AVPR2 (0.38) TP53MAPTALDH1A1GAAMEN1
SCHEMBL8627536 0.77 KCNMA1 (0.35) TP53MAPTKCNMA1ALDH1A1POLB
SCHEMBL8629506 0.77 KCNMA1 (0.36) TP53MAPTKCNMA1ALDH1A1POLB
SCHEMBL8627538 0.76 KCNMA1 (0.36) TP53MAPTKCNMA1ALDH1A1POLB
SCHEMBL8629507 0.76 KCNMA1 (0.36) TP53MAPTKCNMA1ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed