SCHEMBL8628002

SCHEMBL8628002

N#CCn1cc(-c2ccc(Cl)cc2)c(-c2ccccc2S(N)(=O)=O)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.43
PTGS1 P23219 1/20 0.43
F10 P00742 8/20 0.39
F2 P00734 1/20 0.38
PRSS1 P07477 1/20 0.38
PRSS2 P07478 1/20 0.38
PRSS3 P35030 1/20 0.38
CA12 O43570 3/20 0.37
CA1 P00915 3/20 0.37
CA2 P00918 3/20 0.37
CA9 Q16790 3/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.36
RAB9A P51151 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8631526 0.91 ROS1 (0.40) PTGS2F10F2PRSS1PRSS2
SCHEMBL8628932 0.89 ROS1 (0.41) F10F2PRSS1PRSS2PRSS3
SCHEMBL8631613 0.89 PTGS2 (0.43) PTGS2PTGS1F10ALDH1A1MAPT
SCHEMBL8633944 0.86 F10 (0.48) F10F2
SCHEMBL8631834 0.85 PTGS2 (0.46) PTGS2PTGS1F10F2PRSS1
SCHEMBL8629992 0.84 PKM (0.48) PTGS2PTGS1F10F2PRSS1
SCHEMBL7778030 0.84 PTGS2 (0.48) PTGS2PTGS1CA12CA1CA2
SCHEMBL8634432 0.83 PTGS2 (0.44) PTGS2PTGS1F10F2PRSS1
SCHEMBL8635023 0.81 FEN1 (0.44) F10F2PRSS1PRSS2PRSS3
SCHEMBL8627604 0.80 PTGS2 (0.41) PTGS2PTGS1F10F2PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed