SCHEMBL8628003

SCHEMBL8628003

CS(=O)(=O)c1ccc(-c2n[nH]c(OC=O)c2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.49
PTGS1 P23219 5/20 0.49
MAPK11 Q15759 1/20 0.42
MAPK14 Q16539 1/20 0.42
LRRK2 Q5S007 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8629490 0.89 PTGS2 (0.45) PTGS2PTGS1LRRK2
SCHEMBL7779618 0.80 PTGS2 (0.57) PTGS2PTGS1LRRK2
SCHEMBL7779303 0.78 PTGS2 (0.51) PTGS2PTGS1MAPK11MAPK14
SCHEMBL7777645 0.76 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL7778056 0.75 PTGS2 (0.51) PTGS2PTGS1MAPK11MAPK14
SCHEMBL8628027 0.75 GYS1 (0.53) PTGS2PTGS1LRRK2
SCHEMBL7780834 0.75 PTGS2 (0.51) PTGS2PTGS1MAPK11MAPK14
SCHEMBL7772868 0.75 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL8167385 0.75 PTGS2 (0.48) PTGS2PTGS1LRRK2
SCHEMBL7778131 0.74 PTGS2 (0.50) PTGS2PTGS1LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed