SCHEMBL8628397

SCHEMBL8628397

CCC(OC1CCc2cc(F)ccc2N(C(=O)c2ccc([N+](=O)[O-])cc2C)C1)n1ccnc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.33
HTR2C P28335 1/20 0.33
MAPT P10636 4/20 0.32
ALDH1A1 P00352 4/20 0.32
LMNA P02545 2/20 0.32
PDK1 Q15118 4/20 0.32
PDK2 Q15119 4/20 0.32
PDK3 Q15120 4/20 0.32
PDK4 Q16654 4/20 0.32
RAB9A P51151 2/20 0.32
NPC1 O15118 1/20 0.32
POLB P06746 1/20 0.32
THRB P10828 1/20 0.31
MEN1 O00255 1/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
WDR5 P61964 1/20 0.31
HSP90AA1 P07900 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL8634375 0.85 MAPT (0.37) MAPTALDH1A1LMNAPDK1PDK2
SCHEMBL8628399 0.82 ALDH1A1 (0.37) MAPTALDH1A1LMNAMEN1HTT
SCHEMBL8630392 0.81 ALDH1A1 (0.34) MAPTALDH1A1LMNAPDK1PDK2
SCHEMBL8630394 0.75 ALDH1A1 (0.34) MAPTALDH1A1LMNAPDK1PDK2
Iodide SCHEMBL8634376 0.74 KDM4E (0.38) MAPTALDH1A1LMNAPDK1PDK2
SCHEMBL8627671 0.72 AVPR2 (0.37) MAPTALDH1A1LMNARAB9AMEN1
SCHEMBL8628401 0.70 ALDH1A1 (0.37) MAPTALDH1A1LMNAPDK1PDK2
SCHEMBL4682375 0.67 ALDH1A1 (0.38) MAPTALDH1A1LMNAMEN1HTT
SCHEMBL8634457 0.66 TP53 (0.34) MAPTALDH1A1POLBMEN1KMT2A
SCHEMBL8627674 0.66 AVPR2 (0.38) MAPTALDH1A1LMNARAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed