SCHEMBL8628694

SCHEMBL8628694

O=C(O)CNC(=O)c1nc2ccc(S(=O)(=O)c3cc(Cl)cc(Cl)c3)cc2cc1O

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 19/20 0.45
EGLN3 Q9H6Z9 5/20 0.45
FTO Q9C0B1 3/20 0.43
BBOX1 O75936 2/20 0.43
VEGFA P15692 2/20 0.43
FLT1 P17948 2/20 0.43
HIF1AN Q9NWT6 2/20 0.43
TET3 O43151 1/20 0.43
ASPH Q12797 1/20 0.43
TET2 Q6N021 1/20 0.43
KDM8 Q8N371 1/20 0.43
OGFOD1 Q8N543 1/20 0.43
TET1 Q8NFU7 1/20 0.43
KDM5B Q9UGL1 1/20 0.40
KDM2A Q9Y2K7 1/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
THRA P10827 1/20 0.39
THRB P10828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8629264 0.92 EGLN1 (0.51) EGLN1EGLN3FTOBBOX1VEGFA
SCHEMBL8627667 0.92 EGLN1 (0.51) EGLN1EGLN3FTOBBOX1VEGFA
SCHEMBL8629275 0.89 EGLN1 (0.44) EGLN1EGLN3FTOBBOX1VEGFA
SCHEMBL6564105 0.88 EGLN1 (0.48) EGLN1EGLN3FTOBBOX1HIF1AN
SCHEMBL6567419 0.86 EGLN1 (0.51) EGLN1EGLN3FTOHIF1ANKDM5B
SCHEMBL8628250 0.86 EGLN1 (0.46) EGLN1EGLN3FTOHIF1ANKDM5B
SCHEMBL8629451 0.86 EGLN1 (0.55) EGLN1EGLN3FTOHIF1ANKDM5B
SCHEMBL8626818 0.85 EGLN1 (0.44) EGLN1EGLN3FTOBBOX1VEGFA
SCHEMBL8632203 0.84 EGLN1 (0.46) EGLN1EGLN3FTOHIF1ANKDM5B
SCHEMBL8629988 0.83 EGLN1 (0.48) EGLN1FTOHIF1ANTHRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726305-A Substituted quinoline-2-carboxamides, their preparation and their use as pharmaceuticals, and intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-10 US disclosed
US-5719164-A Substituted quinoline-2-carboxamides, their preparation and their use as pharmaceuticals, and intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1998-02-17 US disclosed
EP-0765871-A1 Substituted Quinoline-2-carboxamides, their preparation and their use as prolyle-4-hydroxylase Inhibitors HOECHST AKTIENGESELLSCHAFT (DE) 1997-04-02 EP disclosed