SCHEMBL8629451

SCHEMBL8629451

O=C(O)CNC(=O)c1nc2ccc(S(=O)(=O)c3ccc4ccccc4c3)cc2cc1O

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 14/20 0.55
FTO Q9C0B1 7/20 0.55
HIF1AN Q9NWT6 1/20 0.55
EGLN3 Q9H6Z9 1/20 0.54
KDM5B Q9UGL1 2/20 0.46
KDM2A Q9Y2K7 2/20 0.46
KDM4C Q9H3R0 2/20 0.46
KDM6B O15054 2/20 0.44
KDM3A Q9Y4C1 1/20 0.43
EGLN2 Q96KS0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6564105 0.93 EGLN1 (0.48) EGLN1FTOHIF1ANEGLN3KDM5B
SCHEMBL6567419 0.87 EGLN1 (0.51) EGLN1FTOHIF1ANEGLN3KDM5B
SCHEMBL8629264 0.87 EGLN1 (0.51) EGLN1FTOHIF1ANEGLN3KDM5B
SCHEMBL8628250 0.87 EGLN1 (0.46) EGLN1FTOHIF1ANEGLN3KDM5B
SCHEMBL8628890 0.86 FTO (0.50) EGLN1FTOHIF1ANEGLN3KDM5B
SCHEMBL8629988 0.86 EGLN1 (0.48) EGLN1FTOHIF1AN
SCHEMBL8627667 0.86 EGLN1 (0.51) EGLN1FTOHIF1ANEGLN3KDM5B
SCHEMBL8629275 0.86 EGLN1 (0.44) EGLN1FTOHIF1ANEGLN3KDM5B
SCHEMBL8628694 0.86 EGLN1 (0.45) EGLN1FTOHIF1ANEGLN3KDM5B
SCHEMBL8629876 0.86 EGLN1 (0.51) EGLN1FTOHIF1AN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726305-A Substituted quinoline-2-carboxamides, their preparation and their use as pharmaceuticals, and intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-10 US disclosed
US-5719164-A Substituted quinoline-2-carboxamides, their preparation and their use as pharmaceuticals, and intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1998-02-17 US disclosed
CN-1154365-A Substituted quinoline-2-carboxamides, process for their preparation and their use as pharmaceuticals, and intermediates thereof HOECHST AG (DE) 1997-07-16 CN disclosed
EP-0765871-A1 Substituted Quinoline-2-carboxamides, their preparation and their use as prolyle-4-hydroxylase Inhibitors HOECHST AKTIENGESELLSCHAFT (DE) 1997-04-02 EP disclosed