SCHEMBL8629944

SCHEMBL8629944

NP(N)(=O)NC(=O)c1ccc(C(F)F)s1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.56
HDAC4 P56524 5/20 0.36
HDAC1 Q13547 5/20 0.36
HDAC3 O15379 4/20 0.36
HDAC6 Q9UBN7 5/20 0.35
HPGDS O60760 1/20 0.35
C3AR1 Q16581 3/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HDAC8 Q9BY41 2/20 0.31
CYP2C9 P11712 2/20 0.31
HDAC7 Q8WUI4 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC10 Q969S8 1/20 0.31
HDAC11 Q96DB2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10935147 0.82 HDAC1 (0.43) HDAC4HDAC1HDAC3HDAC6HPGDS
SCHEMBL8630276 0.74 HDAC6 (0.55) HDAC4HDAC1HDAC3HDAC6TAS1R3
SCHEMBL8629681 0.74 F2 (0.57) DAONPC1RAB9AMEN1KMT2A
SCHEMBL8632018 0.74 GAA (0.54) DAONPC1RAB9AMEN1KMT2A
SCHEMBL6375945 0.74 KMT2A (0.53) DAOTAS1R3TAS1R1NPC1RAB9A
SCHEMBL8630679 0.72 DAO (1.00) DAORAB9AMEN1KMT2ACYP2C9
SCHEMBL8629996 0.70 DAO (0.67) DAOHDAC4HDAC1HDAC3HDAC6
SCHEMBL8634109 0.70 SMN1; SMN2 (0.38) HDAC4HDAC1HDAC3HDAC6TAS1R3
SCHEMBL8627366 0.70 SMYD3 (0.54) TAS1R3TAS1R1NPC1RAB9AMEN1
SCHEMBL8628801 0.70 HDAC8 (0.45) HDAC4HDAC1HDAC3HDAC6HPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5840917-A ADMINISTERING TO MAMMAL TO ERADICATE HELICOBACTER PYLORI TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-11-24 US disclosed
WO-1998042347-A1 PHARMACEUTICAL COMPOSITION CONTAINING A PHOSPHORYLAMIDE AND AN AYNTIBIOTIC TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-10-01 WO disclosed
EP-0852498-A1 PHOSPHORYLAMIDES, THEIR PREPARATION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-07-15 EP disclosed
WO-1997011705-A1 PHOSPHORYLAMIDES, THEIR PREPARATION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-04-03 WO disclosed