SCHEMBL8632018

SCHEMBL8632018

NP(N)(=O)NC(=O)c1ccc(Br)s1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
RXFP1 Q9HBX9 1/20 0.54
CES2 O00748 1/20 0.53
CES1 P23141 1/20 0.53
KDM4E B2RXH2 2/20 0.53
ESR1 P03372 1/20 0.53
DAO P14920 1/20 0.52
ALDH1A1 P00352 4/20 0.50
KMT2A Q03164 3/20 0.50
HPGD P15428 3/20 0.50
MEN1 O00255 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.48
GSK3B P49841 2/20 0.47
NPC1 O15118 5/20 0.46
RAB9A P51151 5/20 0.46
MITF O75030 1/20 0.46
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
MAPT P10636 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10935147 0.86 HDAC1 (0.43) GAANPSR1RXFP1KDM4EESR1
SCHEMBL3385006 0.79 GAA (0.65) GAANPSR1RXFP1CES2CES1
SCHEMBL6375945 0.78 KMT2A (0.53) GAANPSR1KDM4EDAOALDH1A1
SCHEMBL8630276 0.78 HDAC6 (0.55) GAARXFP1KDM4EALDH1A1KMT2A
SCHEMBL8629681 0.78 F2 (0.57) NPSR1KDM4EDAOALDH1A1KMT2A
SCHEMBL3848242 0.75 GAA (0.59) GAANPSR1RXFP1CES2CES1
SCHEMBL13753379 0.74 ALDH1A1 (0.63) GAANPSR1RXFP1CES2CES1
SCHEMBL8629944 0.74 DAO (0.56) KDM4EDAOALDH1A1KMT2AHPGD
SCHEMBL8634109 0.74 SMN1; SMN2 (0.38) GAANPSR1KDM4EALDH1A1KMT2A
SCHEMBL8627366 0.74 SMYD3 (0.54) GAAKDM4EALDH1A1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5840917-A ADMINISTERING TO MAMMAL TO ERADICATE HELICOBACTER PYLORI TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-11-24 US disclosed
WO-1998042347-A1 PHARMACEUTICAL COMPOSITION CONTAINING A PHOSPHORYLAMIDE AND AN AYNTIBIOTIC TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-10-01 WO disclosed
EP-0852498-A1 PHOSPHORYLAMIDES, THEIR PREPARATION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-07-15 EP disclosed
WO-1997011705-A1 PHOSPHORYLAMIDES, THEIR PREPARATION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-04-03 WO disclosed