SCHEMBL8630141

SCHEMBL8630141

CNC(=O)CC1CCC(OC)N(C(=O)c2ccc(NC(=O)c3ccccc3C)cc2)c2ccc(F)cc21

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 10/20 0.42
AVPR1A P37288 10/20 0.42
ABCB11 O95342 1/20 0.41
HTR1A P08908 1/20 0.41
CHRM1 P11229 1/20 0.41
OXTR P30559 1/20 0.41
SLC6A4 P31645 1/20 0.41
ADRA1A P35348 1/20 0.41
OPRM1 P35372 1/20 0.41
AVPR1B P47901 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8629514 0.88 AVPR2 (0.44) AVPR2AVPR1AABCB11HTR1ACHRM1
SCHEMBL8635138 0.86 AVPR2 (0.43) AVPR2AVPR1AABCB11HTR1ACHRM1
SCHEMBL8630620 0.86 AVPR1A (0.44) AVPR2AVPR1AABCB11HTR1ACHRM1
SCHEMBL8630121 0.83 NPY2R (0.38) AVPR2AVPR1AABCB11HTR1ACHRM1
SCHEMBL8630730 0.81 AVPR2 (0.47) AVPR2AVPR1AABCB11HTR1ACHRM1
SCHEMBL8631919 0.81 NPY2R (0.39) AVPR2AVPR1AKMT2A
SCHEMBL8627338 0.79 AVPR2 (0.47) AVPR2AVPR1AABCB11HTR1ACHRM1
SCHEMBL8630623 0.78 KMT2A (0.40) KMT2A
Hydrochloric Acid SCHEMBL8634479 0.78 AVPR2 (0.46) AVPR2AVPR1AABCB11HTR1ACHRM1
SCHEMBL8718018 0.77 AVPR2 (0.66) AVPR2AVPR1AABCB11HTR1ACHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed