SCHEMBL8635138

SCHEMBL8635138

COC1CCC(CN2CCN(C)CC2)c2cc(F)ccc2N1C(=O)c1ccc(NC(=O)c2ccccc2C)cc1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 9/20 0.43
AVPR1A P37288 8/20 0.43
OXTR P30559 2/20 0.41
ABCB11 O95342 1/20 0.41
HTR1A P08908 1/20 0.41
CHRM1 P11229 1/20 0.41
SLC6A4 P31645 1/20 0.41
ADRA1A P35348 1/20 0.41
OPRM1 P35372 1/20 0.41
AVPR1B P47901 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8630141 0.86 AVPR2 (0.42) AVPR2AVPR1AOXTRABCB11HTR1A
SCHEMBL8629514 0.85 AVPR2 (0.44) AVPR2AVPR1AOXTRABCB11HTR1A
SCHEMBL8630620 0.82 AVPR1A (0.44) AVPR2AVPR1AOXTRABCB11HTR1A
SCHEMBL8627338 0.81 AVPR2 (0.47) AVPR2AVPR1AABCB11HTR1ACHRM1
SCHEMBL4687543 0.78 AVPR2 (0.54) AVPR2AVPR1AABCB11HTR1ACHRM1
SCHEMBL8631919 0.77 NPY2R (0.39) AVPR2AVPR1A
SCHEMBL8630121 0.77 NPY2R (0.38) AVPR2AVPR1AOXTRABCB11HTR1A
SCHEMBL8630730 0.76 AVPR2 (0.47) AVPR2AVPR1AABCB11HTR1ACHRM1
SCHEMBL8718018 0.76 AVPR2 (0.66) AVPR2AVPR1AOXTRABCB11HTR1A
SCHEMBL8630623 0.75 KMT2A (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed