SCHEMBL8630160

SCHEMBL8630160

CS(=O)(=O)c1ccc(-n2cc(-c3ccc(OC(F)(F)F)cc3)cn2)cc1

nearest known ligand 0.65

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MELK Q14680 2/20 0.65
PTGS2 P35354 14/20 0.55
PTGS1 P23219 8/20 0.46
MAPKAPK2 P49137 1/20 0.46
KIF11 P52732 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7673984 0.81 PTGS2 (0.68) PTGS2PTGS1KIF11
SCHEMBL1228636 0.80 MAPKAPK2 (0.45) MELKMAPKAPK2
SCHEMBL29266901 0.79 ABL1 (0.51) MELKMAPKAPK2
SCHEMBL8631359 0.79 MELK (0.63) MELKPTGS2PTGS1MAPKAPK2KIF11
SCHEMBL182400 0.79 MAPKAPK2 (0.56) MELKMAPKAPK2
SCHEMBL8633662 0.79 MELK (0.76) MELKPTGS2PTGS1
SCHEMBL8630577 0.78 MELK (1.00) MELKPTGS2PTGS1MAPKAPK2
SCHEMBL514383 0.77 PTGS2 (0.65) PTGS2PTGS1KIF11
SCHEMBL23928566 0.76 PTGS2 (0.69) PTGS2
SCHEMBL6290646 0.76 PTGS2 (0.64) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed