SCHEMBL8630229

SCHEMBL8630229

NP(N)(=O)NC(=O)c1sccc1Br

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
GAA P10253 4/20 0.43
KDM4E B2RXH2 3/20 0.43
POLB P06746 1/20 0.42
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
ITGB1 P05556 1/20 0.34
ITGA4 P13612 1/20 0.34
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
CTSL P07711 1/20 0.33
MAPK1 P28482 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1346566 0.79 ALDH1A1 (0.49) ALDH1A1GAAKDM4EPOLBCA12
SCHEMBL8630797 0.79 NPC1 (0.51) GAAKDM4EPOLBKMT2ANPC1
SCHEMBL8633093 0.79 ALDH1A1 (0.36) ALDH1A1GAAKDM4EKMT2AMEN1
SCHEMBL8631451 0.79 GAA (0.51) ALDH1A1GAAPOLBKMT2AMEN1
Hydrochloric Acid SCHEMBL9825967 0.77 KDM4E (0.48) ALDH1A1GAAKDM4EPOLBCA12
SCHEMBL8633756 0.76 KMT2A (0.37) ALDH1A1GAAKDM4EKMT2AMEN1
SCHEMBL8626891 0.75 KMT2A (0.31) ALDH1A1GAAKDM4EKMT2AMEN1
SCHEMBL8630633 0.75 ALDH1A1 (0.40) ALDH1A1GAAKDM4EPOLBKMT2A
SCHEMBL8710088 0.73 NPC1 (0.47) ALDH1A1GAAKDM4EPOLBKMT2A
SCHEMBL13809683 0.73 GAA (0.51) ALDH1A1GAAKDM4EPOLBIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5840917-A ADMINISTERING TO MAMMAL TO ERADICATE HELICOBACTER PYLORI TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-11-24 US disclosed
WO-1998042347-A1 PHARMACEUTICAL COMPOSITION CONTAINING A PHOSPHORYLAMIDE AND AN AYNTIBIOTIC TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-10-01 WO disclosed
EP-0852498-A1 PHOSPHORYLAMIDES, THEIR PREPARATION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-07-15 EP disclosed
WO-1997011705-A1 PHOSPHORYLAMIDES, THEIR PREPARATION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-04-03 WO disclosed