SCHEMBL8633756

SCHEMBL8633756

CCc1ccsc1C(=O)NP(N)(N)=O

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.37
ABCC1 P33527 1/20 0.36
ALDH1A1 P00352 5/20 0.35
MAPT P10636 2/20 0.35
NPC1 O15118 1/20 0.35
PKM P14618 2/20 0.35
GAA P10253 2/20 0.34
GSK3B P49841 1/20 0.34
KDM4E B2RXH2 1/20 0.34
GLA P06280 1/20 0.34
HPGD P15428 1/20 0.34
MAPK1 P28482 1/20 0.34
MEN1 O00255 1/20 0.34
RAB9A P51151 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8630797 0.79 NPC1 (0.51) KMT2AMAPTNPC1PKMGAA
SCHEMBL8631451 0.76 GAA (0.51) KMT2AALDH1A1MAPTNPC1PKM
SCHEMBL8630229 0.76 ALDH1A1 (0.43) KMT2AALDH1A1NPC1GAAKDM4E
SCHEMBL8709676 0.75 PTK2 (0.35) KMT2AABCC1ALDH1A1MAPTNPC1
SCHEMBL2279587 0.74 BCAT2 (0.47) KMT2AABCC1ALDH1A1MAPTNPC1
SCHEMBL8710088 0.74 NPC1 (0.47) KMT2AALDH1A1MAPTNPC1PKM
SCHEMBL2065269 0.72 ABCC1 (0.50) KMT2AABCC1ALDH1A1NPC1GAA
SCHEMBL14614093 0.72 MAPK8 (0.42) KMT2AABCC1ALDH1A1PKMGAA
SCHEMBL8630633 0.72 ALDH1A1 (0.40) KMT2AALDH1A1MAPTNPC1GAA
SCHEMBL8626891 0.72 KMT2A (0.31) KMT2AALDH1A1GAAKDM4EGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5840917-A ADMINISTERING TO MAMMAL TO ERADICATE HELICOBACTER PYLORI TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-11-24 US disclosed
WO-1998042347-A1 PHARMACEUTICAL COMPOSITION CONTAINING A PHOSPHORYLAMIDE AND AN AYNTIBIOTIC TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-10-01 WO disclosed
EP-0852498-A1 PHOSPHORYLAMIDES, THEIR PREPARATION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-07-15 EP disclosed
WO-1997011705-A1 PHOSPHORYLAMIDES, THEIR PREPARATION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-04-03 WO disclosed