SCHEMBL8630565

SCHEMBL8630565

Cc1c(-c2ccc(Cl)cc2)c(-c2ccccc2S(N)(=O)=O)nn1CCc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.40
PTGES2 Q9H7Z7 1/20 0.39
PTGDR2 Q9Y5Y4 2/20 0.39
KDM4E B2RXH2 4/20 0.39
HPGD P15428 4/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
POLB P06746 1/20 0.39
CYP2D6 P10635 1/20 0.39
ADORA2A P29274 1/20 0.39
MAPT P10636 1/20 0.38
TP53 P04637 1/20 0.37
MDM2 Q00987 1/20 0.37
HTR7 P34969 2/20 0.37
HTR1A P08908 1/20 0.37
HTR2A P28223 1/20 0.37
ALDH1A1 P00352 1/20 0.37
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8631591 0.92 PTGS2 (0.41) PTGS2PTGES2KDM4EHPGDCYP3A4
SCHEMBL8631203 0.92 PTGDR2 (0.46) PTGS2PTGDR2KDM4EHPGDCYP3A4
SCHEMBL8632316 0.86 PTGS1 (0.40) PTGS2PTGDR2KDM4EHPGDCYP3A4
SCHEMBL8631669 0.86 PTGES2 (0.38) PTGS2PTGES2KDM4EHPGDCYP3A4
SCHEMBL7779851 0.85 PTGS2 (0.50) PTGS2CYP3A4HTR7HTR1AHTR2A
SCHEMBL8628555 0.85 KDM4E (0.38) PTGS2PTGES2KDM4EHPGDCYP3A4
SCHEMBL8627776 0.85 PTGS2 (0.38) PTGS2PTGES2KDM4EHPGDCYP3A4
SCHEMBL8635575 0.84 PTGS2 (0.46) PTGS2PTGDR2KDM4EHPGDCYP3A4
SCHEMBL8631651 0.84 PTGS2 (0.43) PTGS2PTGES2KDM4EHPGDCYP3A4
SCHEMBL8630965 0.84 PTGS2 (0.47) PTGS2PTGES2KDM4EHPGDCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed