SCHEMBL8628555

SCHEMBL8628555

N#Cc1c(-c2ccc(Cl)cc2)c(-c2ccccc2S(N)(=O)=O)nn1CCc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.38
HPGD P15428 5/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
MAPT P10636 2/20 0.38
PTGES2 Q9H7Z7 1/20 0.38
ALDH1A1 P00352 3/20 0.37
ADORA2A P29274 1/20 0.37
PTGS2 P35354 3/20 0.36
NRP1 O14786 1/20 0.36
POLB P06746 1/20 0.35
CYP2D6 P10635 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
HTT P42858 1/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8631606 0.91 HTR7 (0.39) KDM4EHPGDCYP3A4CYP2C9CYP2C19
SCHEMBL8634745 0.90 PTGS2 (0.38) KDM4EHPGDCYP3A4CYP2C9CYP2C19
SCHEMBL7779758 0.86 PTGS2 (0.46) MAPTPTGS2CA12CA1CA2
SCHEMBL8629956 0.86 PTGS2 (0.37) KDM4EHPGDCYP3A4CYP2C9CYP2C19
SCHEMBL8629352 0.86 F10 (0.38) KDM4EHPGDCYP3A4CYP2C9CYP2C19
SCHEMBL8630565 0.85 PTGS2 (0.40) KDM4EHPGDCYP3A4CYP2C9CYP2C19
SCHEMBL8631669 0.83 PTGES2 (0.38) KDM4EHPGDCYP3A4CYP2C9CYP2C19
SCHEMBL8627776 0.83 PTGS2 (0.38) KDM4EHPGDCYP3A4CYP2C9CYP2C19
SCHEMBL8635045 0.82 PDE9A (0.42) KDM4EHPGDCYP3A4CYP2C9CYP2C19
SCHEMBL8634717 0.82 PTGS2 (0.43) PTGS2F10PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed