SCHEMBL8631463

SCHEMBL8631463

NP(N)(=O)NC(=O)c1cc(Cl)c(Cl)s1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 2/20 0.53
GSK3B P49841 1/20 0.49
HDAC3 O15379 2/20 0.35
HDAC4 P56524 2/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC7 Q8WUI4 2/20 0.35
HDAC2 Q92769 2/20 0.35
HDAC10 Q969S8 2/20 0.35
HDAC11 Q96DB2 2/20 0.35
HDAC8 Q9BY41 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
HDAC9 Q9UKV0 2/20 0.35
HDAC5 Q9UQL6 2/20 0.35
CYP2D6 P10635 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
ABL1 P00519 1/20 0.31
ALDH1A1 P00352 2/20 0.31
GAA P10253 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8633480 0.83 DAO (0.56) DAOGSK3BHDAC3HDAC4HDAC1
SCHEMBL8630205 0.83 ALDH1A1 (0.37) DAOGSK3BHDAC3HDAC4HDAC1
SCHEMBL8629681 0.73 F2 (0.57) DAOGSK3BALDH1A1KDM4E
SCHEMBL8634421 0.73 DAO (0.55) DAOGSK3BKDM4E
SCHEMBL10935147 0.72 HDAC1 (0.43) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL5009880 0.72 DAO (0.65) DAOGSK3BCYP2D6SLC6A2SLC6A4
SCHEMBL8627665 0.71 MEN1 (0.53) GSK3BALDH1A1KDM4E
SCHEMBL8633709 0.71 ALDH1A1 (0.41) GSK3BALDH1A1GAA
SCHEMBL8634456 0.70 MAPT (0.41) DAOGSK3BALDH1A1GAAKDM4E
SCHEMBL21612137 0.70 DAO (0.56) DAOGSK3BKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5840917-A ADMINISTERING TO MAMMAL TO ERADICATE HELICOBACTER PYLORI TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-11-24 US disclosed
EP-0852498-A1 PHOSPHORYLAMIDES, THEIR PREPARATION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-07-15 EP disclosed
WO-1997011705-A1 PHOSPHORYLAMIDES, THEIR PREPARATION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-04-03 WO disclosed