SCHEMBL8631478

SCHEMBL8631478

c1ccc2c(c1)cnn2CN1CCN(Cc2ccc3c(c2)OCO3)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
KDM4E B2RXH2 3/20 0.54
POLB P06746 1/20 0.54
CYP2D6 P10635 3/20 0.53
MEN1 O00255 2/20 0.53
CYP1A2 P05177 2/20 0.53
CYP3A4 P08684 2/20 0.53
CYP2C19 P33261 2/20 0.53
KMT2A Q03164 2/20 0.53
USP2 O75604 1/20 0.53
HTR1A P08908 1/20 0.53
ADRA2A P08913 1/20 0.53
DRD2 P14416 1/20 0.53
ADRA2B P18089 1/20 0.53
ADRA2C P18825 1/20 0.53
NFKB1 P19838 1/20 0.53
SLC6A2 P23975 1/20 0.53
MAPK1 P28482 1/20 0.53
SLC6A4 P31645 1/20 0.53
ADRA1A P35348 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8631501 0.84 SLC6A4 (0.44) ALDH1A1KDM4EPOLBCYP2D6MEN1
SCHEMBL8631008 0.80 RECQL (0.67) ALDH1A1POLBKMT2AHTR1AADRA2A
SCHEMBL108678 0.77 KDM4E (0.70) KDM4ECYP2D6MEN1CYP1A2CYP3A4
SCHEMBL2316901 0.76 CYP2D6 (0.82) ALDH1A1KDM4ECYP2D6MEN1CYP1A2
SCHEMBL10833328 0.74 KDM4E (0.71) ALDH1A1KDM4EPOLBCYP2D6MEN1
SCHEMBL29520874 0.73 RECQL (0.53) POLBCYP2D6CYP1A2ADRA2AHSD17B10
SCHEMBL6977835 0.72 RECQL (0.51) POLBCYP1A2ADRA2AHSD17B10TSHR
SCHEMBL4750999 0.71 HTR2B (0.67) ALDH1A1KDM4EHTR1ADRD2HTR2B
SCHEMBL12237371 0.71 KDM4E (0.76) ALDH1A1KDM4EPOLBCYP2D6MEN1
SCHEMBL6231529 0.71 KDM4E (0.74) ALDH1A1KDM4EPOLBCYP2D6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780475-A Antipsychotic indazole derivatives MERCK, SHARP & DOHME LIMITED (GB) 1998-07-14 US disclosed