SCHEMBL8631944

SCHEMBL8631944

C#CCn1nc(NS(=O)(=O)c2ccccc2)c(-c2ccc(OC)cc2)c1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.44
GAA P10253 1/20 0.44
ALDH1A1 P00352 2/20 0.40
GGT1 P19440 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
MAPT P10636 4/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
ADORA1 P30542 1/20 0.39
PPARG P37231 1/20 0.39
NPY5R Q15761 1/20 0.38
POLB P06746 1/20 0.38
MEN1 O00255 2/20 0.38
STAT3 P40763 1/20 0.38
PKM P14618 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
LMNA P02545 3/20 0.38
TP53 P04637 1/20 0.38
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8631393 0.91 KMT2A (0.42) KMT2AGAAALDH1A1GGT1PTGDR2
SCHEMBL8631537 0.90 EDNRB (0.41) KMT2AALDH1A1MAPTSMN1; SMN2PPARG
SCHEMBL8630980 0.89 KMT2A (0.39) KMT2AALDH1A1MAPTSMN1; SMN2TDP1
SCHEMBL8634609 0.88 KMT2A (0.45) KMT2AGAAALDH1A1GGT1PTGDR2
SCHEMBL8628674 0.88 PTGS2 (0.44) KMT2AMAPTPOLBMEN1NPSR1
SCHEMBL8630567 0.87 EDNRB (0.41) KMT2AALDH1A1PTGDR2MAPTPOLB
SCHEMBL8629114 0.87 ALDH1A1 (0.36) KMT2AGAAALDH1A1MAPTSMN1; SMN2
SCHEMBL8629013 0.87 PPARA (0.39) MAPTCYP2C9
SCHEMBL8627950 0.87 MAPT (0.38) KMT2AALDH1A1MAPTSMN1; SMN2POLB
SCHEMBL8631438 0.87 CYP1A2 (0.46) KMT2AGAAALDH1A1GGT1PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed