SCHEMBL8631945

SCHEMBL8631945

CCCCCCN1c2ccccc2Sc2c(CN3C(=O)c4ccc(C(O[SiH2]C(C)(C)C)(c5ccccc5)c5ccccc5)cc4C3=O)cccc21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDF Q9HBH1 1/20 0.34
CDC25A P30304 4/20 0.33
CES1 P23141 2/20 0.33
FPR2 P25090 3/20 0.33
HDAC6 Q9UBN7 3/20 0.33
HDAC3 O15379 2/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC7 Q8WUI4 2/20 0.33
HDAC2 Q92769 2/20 0.33
HDAC9 Q9UKV0 2/20 0.33
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
TP53 P04637 2/20 0.33
NPC1 O15118 1/20 0.33
ABCB11 O95342 1/20 0.33
CYP1A2 P05177 1/20 0.33
CHRM2 P08172 1/20 0.33
ABCB1 P08183 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8632480 0.88 HPGD (0.34) TP53ADRA2ASLC6A2SLC6A4DRD3
SCHEMBL7392961 0.85 CDC25A (0.38) CDC25ACES1BCHEACHEALDH1A1
SCHEMBL7390458 0.80 PDF (0.39) PDFFPR2HDAC6TP53NPC1
SCHEMBL8630694 0.79 HPGD (0.35) TP53ADRA2ASLC6A2SLC6A4DRD3
SCHEMBL8631941 0.77 PDF (0.33) PDFCDC25ACES1HDAC6HDAC3
SCHEMBL7386866 0.74 PDF (0.32) PDFCDC25ACES1
SCHEMBL7398242 0.73 GAA (0.33) CYP1A2CHRM2HTR1AADRA2ATSHR
SCHEMBL7392958 0.70 CDC25A (0.39) CDC25ACES1ACHETSHRALDH1A1
SCHEMBL7391109 0.70 CDC25A (0.46) CDC25ACES1ACHEMAPTALDH1A1
SCHEMBL7392955 0.69 CDC25A (0.37) CDC25ACES1BCHEACHETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5811548-A USEFUL AS RESEARCH TOOLS IN THE DETERMINATION OF BIOLOGICALLY ACTIVE PEPTIDE SEQUENCES HOFFMANN-LA ROCHE INC. (US) 1998-09-22 US disclosed
US-5811389-A INHIBITING PLATELET AGGREGATION; BLOOD DISORDERS HOFFMANN-LA ROCHE INC. (US) 1998-09-22 US disclosed