SCHEMBL8631941

SCHEMBL8631941

CCCCCCN1c2ccccc2Sc2c(CN3C(=O)c4ccc(CO[Si](c5ccccc5)(c5ccccc5)C(C)(C)C)cc4C3=O)cccc21

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDF Q9HBH1 2/20 0.33
CDC25A P30304 10/20 0.32
CES1 P23141 2/20 0.32
HDAC3 O15379 2/20 0.32
HDAC1 Q13547 2/20 0.32
HDAC7 Q8WUI4 2/20 0.32
HDAC2 Q92769 2/20 0.32
HDAC6 Q9UBN7 2/20 0.32
HDAC9 Q9UKV0 2/20 0.32
PDCD1 Q15116 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
TUBB4A P04350 1/20 0.31
TUBB P07437 1/20 0.31
TUBA3C P0DPH7 1/20 0.31
HDAC4 P56524 1/20 0.31
TUBA1B P68363 1/20 0.31
TUBA4A P68366 1/20 0.31
TUBB4B P68371 1/20 0.31
TUBB3 Q13509 1/20 0.31
TUBB2A Q13885 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8632477 0.88 PDCD1 (0.35) HDAC3HDAC1HDAC7HDAC2HDAC6
SCHEMBL7392958 0.87 CDC25A (0.39) CDC25ACES1ALDH1A1ALDH2ALDH3A1
SCHEMBL7390456 0.84 PDF (0.39) PDFHDAC6ALDH1A1LMNAMEN1
SCHEMBL8630691 0.78 PDCD1 (0.35) PDCD1CD274LMNAMEN1HPGD
SCHEMBL8631945 0.77 PDF (0.34) PDFCDC25ACES1HDAC3HDAC1
SCHEMBL7398238 0.75 GAA (0.34) LMNAMEN1TSHRRECQLKMT2A
SCHEMBL7386864 0.74 TLR8 (0.33) PDFCDC25AALDH1A1MEN1KMT2A
SCHEMBL8630245 0.73 PDF (0.33) PDFCDC25ACES1MEN1KMT2A
SCHEMBL8627860 0.72 MEN1 (0.31) ALDH1A1MEN1KMT2A
SCHEMBL7431775 0.69 MAOA (0.41) ALDH1A1LMNAMEN1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5811548-A USEFUL AS RESEARCH TOOLS IN THE DETERMINATION OF BIOLOGICALLY ACTIVE PEPTIDE SEQUENCES HOFFMANN-LA ROCHE INC. (US) 1998-09-22 US disclosed
US-5811389-A INHIBITING PLATELET AGGREGATION; BLOOD DISORDERS HOFFMANN-LA ROCHE INC. (US) 1998-09-22 US disclosed