SCHEMBL8632045

SCHEMBL8632045

COCCN(C(C)=O)C(=O)C(Oc1ccccc1)N1CCN(c2ccncc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.42
TP53 P04637 2/20 0.40
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40
HRH3 Q9Y5N1 4/20 0.40
TSHR P16473 3/20 0.40
ALDH1A1 P00352 3/20 0.40
GAA P10253 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
NPY2R P49146 1/20 0.40
KDM4E B2RXH2 2/20 0.39
RORC P51449 1/20 0.39
MAPT P10636 1/20 0.39
HRH2 P25021 1/20 0.39
HRH1 P35367 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
MAPK1 P28482 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HIF1A Q16665 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8636543 0.87 ITGB3 (0.41) ROCK2TP53ITGB3ITGA2BHRH3
SCHEMBL8632702 0.83 ROCK2 (0.44) ROCK2TP53ITGB3ITGA2BHRH3
SCHEMBL8696501 0.78 CYP2C9 (0.49) ROCK2ITGB3ITGA2BHRH3TSHR
SCHEMBL8633635 0.77 TSHR (0.44) ROCK2TP53ITGB3ITGA2BHRH3
Hydrochloric Acid SCHEMBL8637477 0.76 GAA (0.46) ROCK2TP53ITGB3ITGA2BHRH3
SCHEMBL8634059 0.75 ITGB3 (0.44) ROCK2TP53ITGB3ITGA2BHRH3
Hydrochloric Acid SCHEMBL8699382 0.74 ITGB3 (0.43) ROCK2TP53ITGB3ITGA2BHRH3
SCHEMBL8636921 0.73 SMN1; SMN2 (0.42) ROCK2TP53ITGB3ITGA2BHRH3
SCHEMBL8633547 0.72 TSHR (0.42) ROCK2TP53ITGB3ITGA2BHRH3
SCHEMBL8632821 0.70 ITGB3 (0.47) ROCK2TP53ITGB3ITGA2BHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed