SCHEMBL8633635

SCHEMBL8633635

CC(=O)OC(=O)C(Oc1ccccc1)N1CCN(c2ccncc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.44
CYP2C9 P11712 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
ALDH1A1 P00352 2/20 0.44
CYP2D6 P10635 1/20 0.44
MAPK1 P28482 1/20 0.44
HIF1A Q16665 1/20 0.44
ITGB3 P05106 1/20 0.43
ITGA2B P08514 1/20 0.43
ROCK2 O75116 1/20 0.43
GAA P10253 3/20 0.41
KDM4E B2RXH2 2/20 0.41
MAPT P10636 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
HRH3 Q9Y5N1 5/20 0.40
NPY2R P49146 1/20 0.40
HRH2 P25021 1/20 0.39
HRH1 P35367 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634059 0.89 ITGB3 (0.44) TSHRCYP2C9SMN1; SMN2ALDH1A1CYP2D6
Hydrochloric Acid SCHEMBL8699382 0.88 ITGB3 (0.43) TSHRCYP2C9SMN1; SMN2ALDH1A1CYP2D6
SCHEMBL8700994 0.86 AOC3 (0.41) TSHRALDH1A1MAPK1MAPTHSD17B10
SCHEMBL8633385 0.85 HSD17B10 (0.43) TSHRSMN1; SMN2ALDH1A1MAPK1ROCK2
SCHEMBL8696501 0.85 CYP2C9 (0.49) TSHRCYP2C9SMN1; SMN2ALDH1A1CYP2D6
Hydrochloric Acid SCHEMBL8637477 0.85 GAA (0.46) TSHRCYP2C9SMN1; SMN2ALDH1A1CYP2D6
SCHEMBL8633823 0.84 NCF1 (0.39) TSHRALDH1A1MAPK1KDM4EMAPT
SCHEMBL8696260 0.84 CYP2C9 (0.38) TSHRCYP2C9SMN1; SMN2ALDH1A1CYP2D6
Hydrochloric Acid SCHEMBL8631358 0.83 CYP2C9 (0.38) TSHRCYP2C9SMN1; SMN2ALDH1A1CYP2D6
SCHEMBL8635654 0.83 MAPT (0.44) TSHRALDH1A1MAPK1ROCK2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed