SCHEMBL8632051

SCHEMBL8632051

COCCNC(=O)C(Oc1ccccc1)(C(C)=O)N1CCN(c2ccncc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HRH3 Q9Y5N1 5/20 0.39
KMT2A Q03164 2/20 0.39
DRD4 P21917 2/20 0.39
HRH2 P25021 1/20 0.38
HRH1 P35367 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HIF1A Q16665 1/20 0.38
DRD2 P14416 1/20 0.38
F10 P00742 1/20 0.38
MAPT P10636 1/20 0.38
MEN1 O00255 1/20 0.38
PLA2G1B P04054 1/20 0.38
ATG4B Q9Y4P1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8698910 0.90 HRH3 (0.40) HRH3DRD4HRH2HRH1ALDH1A1
SCHEMBL8636548 0.86 GFER (0.42) HTR2AHTR2CHRH3ALDH1A1MAPK1
SCHEMBL8632705 0.85 CYP2C9 (0.42) HRH3HRH2HRH1ALDH1A1CYP2D6
SCHEMBL8633634 0.82 CYP2C9 (0.46) HRH3HRH2HRH1ALDH1A1CYP2D6
SCHEMBL8635264 0.80 CYP2C9 (0.44) HRH3HRH2HRH1ALDH1A1CYP2D6
SCHEMBL8634057 0.75 CYP2C9 (0.43) HRH3HRH2HRH1ALDH1A1CYP2D6
SCHEMBL8635770 0.75 ROCK2 (0.49) KMT2ADRD4ALDH1A1CYP2D6CYP2C9
SCHEMBL8632213 0.74 SLC2A1 (0.43) KMT2AALDH1A1TSHRHIF1AF10
Hydrochloric Acid SCHEMBL8636995 0.74 CYP2C9 (0.42) HRH3HRH2HRH1ALDH1A1CYP2D6
SCHEMBL8630430 0.73 ITGB3 (0.45) HRH3HRH2HRH1ALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed