SCHEMBL8632213

SCHEMBL8632213

COc1ccccc1OC(C(C)=O)(C(=O)O)N1CCN(c2ccncc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
GAA P10253 2/20 0.40
ALDH1A1 P00352 2/20 0.40
TSHR P16473 1/20 0.40
HTR1A P08908 1/20 0.40
ADRA1A P35348 1/20 0.40
TP53 P04637 2/20 0.40
GFER P55789 2/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 4/20 0.39
KDM4E B2RXH2 2/20 0.39
TYR P14679 1/20 0.39
KHK P50053 1/20 0.39
CHRM1 P11229 1/20 0.39
F10 P00742 1/20 0.38
RAB9A P51151 1/20 0.38
LMNA P02545 1/20 0.38
HIF1A Q16665 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634909 0.89 KDM4E (0.39) SLC2A1GAAALDH1A1TSHRMAPT
SCHEMBL8635651 0.87 ALDH1A1 (0.46) MEN1KMT2AGAAALDH1A1TSHR
SCHEMBL8633634 0.86 CYP2C9 (0.46) GAAALDH1A1TSHRMAPTKDM4E
SCHEMBL8635770 0.83 ROCK2 (0.49) KMT2AGAAALDH1A1TSHRTP53
SCHEMBL8636233 0.80 CHRM1 (0.39) SLC2A1GAATSHRMAPTKDM4E
SCHEMBL8635264 0.80 CYP2C9 (0.44) GAAALDH1A1TSHRMAPTKDM4E
SCHEMBL8634772 0.79 GAA (0.39) GAAALDH1A1TSHRMAPTKDM4E
SCHEMBL8631971 0.78 ITGB3 (0.40) SLC2A1MEN1KMT2AGAAALDH1A1
SCHEMBL8698910 0.76 HRH3 (0.40) GAAALDH1A1TSHRTP53MAPT
SCHEMBL8632705 0.76 CYP2C9 (0.42) GAAALDH1A1TSHRMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed