SCHEMBL8632180

SCHEMBL8632180

CC(=O)N(Cc1ccccc1)Oc1ccc(C(=O)CBr)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 5/20 0.49
PTPN1 P18031 4/20 0.47
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
ACHE P22303 2/20 0.43
ALOX5 P09917 1/20 0.43
PTGS1 P23219 1/20 0.43
PTGS2 P35354 1/20 0.43
MAOB P27338 1/20 0.41
EGFR P00533 2/20 0.41
ALDH1A1 P00352 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6957841 0.80 ALOX5 (0.47) NPC1RAB9AACHEALOX5PTGS1
SCHEMBL6965769 0.76 ALDH1A1 (0.57) MAOBALDH1A1CYP2C9CYP2C19L3MBTL1
SCHEMBL14087168 0.76 ACHE (0.52) GSK3BPTPN1NPC1RAB9AACHE
SCHEMBL4877516 0.74 TSHR (0.63) ACHEMAOBEGFRALDH1A1MEN1
SCHEMBL10506729 0.73 GSK3B (0.55) GSK3BPTPN1NPC1RAB9AALDH1A1
SCHEMBL41220 0.72 NR4A1 (0.70) GSK3BPTPN1RAB9APTGS1PTGS2
SCHEMBL6326282 0.72 BCHE (0.48) GSK3BPTPN1NPC1RAB9AACHE
SCHEMBL1350830 0.71 GSK3B (0.67) GSK3BPTPN1
SCHEMBL27862677 0.71 ALOX5 (0.47) NPC1RAB9AACHEALOX5PTGS1
SCHEMBL2531747 0.69 GSK3B (0.69) GSK3BPTPN1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed