SCHEMBL8632723

SCHEMBL8632723

CCCCOC(C)(C(=O)OC1CCN(c2ccncc2)CC1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 3/20 0.49
MLNR O43193 1/20 0.49
CHRM2 P08172 1/20 0.49
CHRM1 P11229 1/20 0.49
HTR2A P28223 1/20 0.49
HTR2C P28335 1/20 0.49
HRH1 P35367 1/20 0.49
OPRM1 P35372 1/20 0.49
DRD3 P35462 1/20 0.49
OPRK1 P41145 1/20 0.49
HTR2B P41595 1/20 0.49
SLC6A3 Q01959 1/20 0.49
KCNH2 Q12809 1/20 0.49
CACNA1C Q13936 1/20 0.49
HRH3 Q9Y5N1 3/20 0.44
LSS P48449 1/20 0.40
CYP19A1 P11511 1/20 0.40
ITGB3 P05106 2/20 0.39
ITGA2B P08514 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8605444 0.71 HRH3 (0.56) HRH3CYP19A1ITGB3ITGA2B
SCHEMBL27967028 0.71 GPR119 (0.53) CHRM3MLNRCHRM2CHRM1HTR2A
SCHEMBL7401896 0.69 HRH3 (0.62) HRH3LSSITGB3ITGA2B
SCHEMBL27663466 0.69 TSHR (0.45) CHRM3MLNRCHRM2CHRM1HTR2A
Hydrochloric Acid SCHEMBL6207497 0.68 HRH3 (0.61) HRH3LSSITGB3ITGA2B
SCHEMBL8632715 0.68 HRH3 (0.43) HRH1HRH3ITGB3ITGA2B
SCHEMBL8633871 0.67 CYP2C9 (0.53) HRH3LSSITGB3ITGA2B
Hydrochloric Acid SCHEMBL8632011 0.67 HRH3 (0.60) HRH3LSSITGB3ITGA2B
Propiverine SCHEMBL14672394 0.67 CHRM3 (0.95) CHRM3MLNRCHRM2CHRM1HTR2A
SCHEMBL8632718 0.67 CYP2C9 (0.45) HRH1HRH3ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed