SCHEMBL8632715

SCHEMBL8632715

CCCCOc1ccccc1OC(=O)C(C)C1CCN(c2ccncc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 8/20 0.43
SPHK1 Q9NYA1 2/20 0.42
CCNC P24863 1/20 0.42
CDK8 P49336 1/20 0.42
ITGB3 P05106 3/20 0.42
ITGA2B P08514 3/20 0.42
F10 P00742 5/20 0.41
HRH1 P35367 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8637462 0.78 HRH3 (0.42) HRH3CCNCCDK8F10
SCHEMBL8637204 0.75 HRH3 (0.44) HRH3CCNCCDK8ITGB3ITGA2B
SCHEMBL8632718 0.72 CYP2C9 (0.45) HRH3SPHK1CCNCCDK8ITGB3
SCHEMBL6160214 0.71 SPHK1 (0.46) HRH3SPHK1ITGB3ITGA2B
SCHEMBL21385141 0.70 MAPT (0.45)
SCHEMBL8683270 0.69 F10 (0.44) HRH3CCNCCDK8ITGB3ITGA2B
SCHEMBL8632723 0.68 CHRM3 (0.49) HRH3ITGB3ITGA2BHRH1
SCHEMBL7334680 0.68 CHKA (0.52) HRH3ITGB3ITGA2B
SCHEMBL7334443 0.67 SMN1; SMN2 (0.56)
SCHEMBL8632780 0.67 F10 (0.45) HRH3F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed