SCHEMBL8633208

SCHEMBL8633208

O=S(=O)(Nc1nn(CCCO)c(C(F)(F)F)c1-c1ccc(Cl)cc1)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 3/20 0.46
EDNRA P25101 3/20 0.46
KDM1A O60341 5/20 0.40
PTGS2 P35354 2/20 0.39
MALT1 Q9UDY8 2/20 0.37
ERBB2 P04626 1/20 0.37
HSP90AA1 P07900 1/20 0.37
HSP90AB1 P08238 1/20 0.37
MAPT P10636 2/20 0.36
NAT1 P18440 1/20 0.36
PTGES O14684 1/20 0.36
ALOX5 P09917 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8631638 0.93 EDNRB (0.47) EDNRBEDNRAPTGS2MAPTALDH1A1
SCHEMBL8627989 0.91 PTGS2 (0.48) EDNRBEDNRAPTGS2MAPTALDH1A1
SCHEMBL8633251 0.90 EDNRA (0.41) EDNRBEDNRAPTGS2MALT1MAPT
SCHEMBL8632637 0.88 EDNRB (0.40) EDNRBEDNRAPTGS2MAPTALDH1A1
SCHEMBL8631658 0.88 EDNRB (0.42) EDNRBEDNRAPTGS2MAPTALDH1A1
SCHEMBL8631240 0.87 ERBB2 (0.39) EDNRBEDNRAPTGS2MALT1ERBB2
SCHEMBL8629982 0.86 EDNRB (0.43) EDNRBEDNRAKDM1APTGS2MAPT
SCHEMBL8630539 0.86 PTGS2 (0.46) EDNRBEDNRAKDM1APTGS2MAPT
SCHEMBL8631938 0.85 ALDH1A1 (0.41) EDNRBEDNRAKDM1APTGS2MAPT
SCHEMBL8631961 0.84 PTGS2 (0.38) EDNRBEDNRAPTGS2MALT1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed