SCHEMBL8633347

SCHEMBL8633347

Cc1ncsc1C(O)c1cccs1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.44
MAPT P10636 3/20 0.43
HSD17B10 Q99714 1/20 0.43
IDO1 P14902 4/20 0.42
TDO2 P48775 4/20 0.42
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
CNR2 P34972 1/20 0.39
TOP2A P11388 2/20 0.38
TOP2B Q02880 2/20 0.38
EGFR P00533 1/20 0.38
PKM P14618 2/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38
ATM Q13315 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8683323 0.80 KDM4E (0.43) PKMALDH1A1KMT2AKDM4EP2RX7
SCHEMBL9051451 0.80 KDM4E (0.38) TSHRMAPTHSD17B10IDO1TDO2
SCHEMBL2593085 0.76 SLC6A3 (0.44) IDO1TDO2PKMALDH1A1HPGD
SCHEMBL8633179 0.75 CYP3A4 (0.40) TSHRMAPTHSD17B10PKMALDH1A1
SCHEMBL8634063 0.73 FFAR2 (0.38) PKMALDH1A1HPGDKMT2AKDM4E
SCHEMBL8629570 0.73 GAA (0.44) MAPTIDO1TDO2PKMALDH1A1
SCHEMBL1384962 0.73 TSHR (0.57) TSHRMAPTHSD17B10IDO1TDO2
SCHEMBL9051447 0.73 CYP2C19 (0.42) TSHRMAPTRAB9AALDH1A1HPGD
SCHEMBL8631255 0.72 KMT2A (0.36) MAPTHSD17B10PKMALDH1A1L3MBTL1
Hydrochloric Acid SCHEMBL9046489 0.72 KMT2A (0.39) TSHRMAPTHSD17B10IDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5712299-A TREATMENT OF NEURODEGENERATIVE DISORDERS ASTRA AKTIEBOLAG (SE) 1998-01-27 US claimed
EP-0707574-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES Astra Aktiebolag (SE) 1996-04-24 EP claimed
WO-1995001968-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES ASTRA AKTIEBOLAG (SE) 1995-01-19 WO claimed
US-5712299-A TREATMENT OF NEURODEGENERATIVE DISORDERS ASTRA AKTIEBOLAG (SE) 1998-01-27 US disclosed
EP-0707574-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES Astra Aktiebolag (SE) 1996-04-24 EP disclosed
WO-1995001968-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES ASTRA AKTIEBOLAG (SE) 1995-01-19 WO disclosed