SCHEMBL8629570

SCHEMBL8629570

Cc1ccccc1C(O)c1scnc1C

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.44
P2RX7 Q99572 3/20 0.36
ESR1 P03372 1/20 0.36
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
SLC6A3 Q01959 1/20 0.33
KDM4E B2RXH2 1/20 0.33
PKM P14618 1/20 0.33
ACP3 P15309 1/20 0.33
CTSA P10619 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
KMT2A Q03164 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
CHEK2 O96017 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8633796 0.84 ADRB2 (0.36) P2RX7IDO1TDO2SLC6A3
SCHEMBL8629431 0.84 BRD4 (0.39) P2RX7IDO1TDO2
SCHEMBL8629520 0.83 ACHE (0.44) IDO1TDO2ALDH1A1LMNAMAPT
SCHEMBL8630486 0.81 KMT2A (0.46) GAAALDH1A1LMNAMAPTKMT2A
SCHEMBL8683323 0.80 KDM4E (0.43) P2RX7SLC6A3KDM4EPKMMEN1
SCHEMBL2593085 0.79 SLC6A3 (0.44) IDO1TDO2SLC6A3KDM4EPKM
SCHEMBL9525798 0.77 GAA (0.44) GAAESR1IDO1TDO2ACP3
SCHEMBL8633347 0.73 TSHR (0.44) P2RX7IDO1TDO2KDM4EPKM
SCHEMBL598722 0.73 GAA (0.57) GAAESR1IDO1TDO2SLC6A3
SCHEMBL8631255 0.72 KMT2A (0.36) P2RX7KDM4EPKMMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5712299-A TREATMENT OF NEURODEGENERATIVE DISORDERS ASTRA AKTIEBOLAG (SE) 1998-01-27 US disclosed
EP-0707574-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES Astra Aktiebolag (SE) 1996-04-24 EP disclosed
WO-1995001968-A1 NOVEL (1-PHENYL-1-HETEROCYCLYL)METHANOL AND (1-PHENYL-1-HETEROCYCLYL)METHYLAMINE DERIVATIVES ASTRA AKTIEBOLAG (SE) 1995-01-19 WO disclosed