SCHEMBL8633371

SCHEMBL8633371

Cc1ccc(S(=O)(=O)OC(C)OC2CCCc3cc(Cl)ccc3N2C(=O)c2ccc(N)cc2C)cc1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 3/20 0.49
MAPT P10636 2/20 0.35
PDK1 Q15118 4/20 0.33
PDK2 Q15119 4/20 0.33
PDK3 Q15120 4/20 0.33
PDK4 Q16654 4/20 0.33
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
CCR8 P51685 1/20 0.32
BCL2L1 Q07817 1/20 0.32
MCL1 Q07820 1/20 0.32
KMT2A Q03164 1/20 0.32
THRB P10828 1/20 0.32
HTT P42858 1/20 0.31
NPY5R Q15761 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8627187 0.92 AVPR2 (0.40) AVPR2MAPTTP53KMT2A
SCHEMBL8627398 0.89 AVPR2 (0.37) AVPR2MAPTLMNAKMT2AHTT
SCHEMBL8634667 0.88 AVPR2 (0.51) AVPR2MAPTPDK1PDK2PDK3
SCHEMBL8633374 0.85 AVPR2 (0.52) AVPR2MAPTPDK1PDK2PDK3
SCHEMBL8629474 0.84 AVPR2 (0.51) AVPR2MAPTPDK1PDK2PDK3
SCHEMBL8630162 0.83 TSHR (0.38) MAPTPDK1PDK2PDK3PDK4
SCHEMBL8627536 0.82 KCNMA1 (0.35) MAPTLMNATP53KMT2AHTT
SCHEMBL8634668 0.81 AVPR2 (0.51) AVPR2MAPTPDK1PDK2PDK3
SCHEMBL8630766 0.79 AVPR2 (0.41) AVPR2MAPTTP53KMT2A
SCHEMBL8627190 0.77 AVPR2 (0.42) AVPR2MAPTTP53KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed