SCHEMBL8634668

SCHEMBL8634668

Cc1ccc(S(=O)(=O)OCCC2CCCc3cc(Cl)ccc3N2C(=O)c2ccc(N)cc2C)cc1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 2/20 0.51
MAPT P10636 2/20 0.36
CASP3 P42574 3/20 0.35
CASP7 P55210 3/20 0.35
THRB P10828 1/20 0.34
APP P05067 2/20 0.33
LMNA P02545 2/20 0.33
TP53 P04637 2/20 0.33
PDK1 Q15118 2/20 0.33
PDK2 Q15119 2/20 0.33
PDK3 Q15120 2/20 0.33
PDK4 Q16654 2/20 0.33
BCL2L1 Q07817 1/20 0.33
MCL1 Q07820 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8630767 0.92 AVPR2 (0.41) AVPR2MAPTCASP3CASP7TP53
SCHEMBL8630680 0.88 AVPR2 (0.38) AVPR2MAPTCASP3CASP7LMNA
SCHEMBL8633374 0.88 AVPR2 (0.52) AVPR2MAPTTHRBLMNATP53
SCHEMBL8629474 0.87 AVPR2 (0.51) AVPR2MAPTCASP3CASP7THRB
SCHEMBL8632674 0.85 AVPR2 (0.51) AVPR2MAPTLMNATP53
SCHEMBL8634667 0.82 AVPR2 (0.51) AVPR2MAPTTHRBLMNATP53
SCHEMBL8629507 0.82 KCNMA1 (0.36) MAPTCASP3CASP7LMNATP53
SCHEMBL8633371 0.81 AVPR2 (0.49) AVPR2MAPTTHRBLMNATP53
SCHEMBL8627190 0.80 AVPR2 (0.42) AVPR2MAPTTP53KMT2A
SCHEMBL4684422 0.79 AVPR2 (0.51) AVPR2CASP3CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed