SCHEMBL8634182

SCHEMBL8634182

c1ccc(OCN2CCN(c3ccncc3)CC2)cc1

nearest known ligand 0.65

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 14/20 0.65
HRH1 P35367 9/20 0.65
HRH2 P25021 5/20 0.65
HTR1A P08908 2/20 0.55
DRD2 P14416 2/20 0.55
HTR2A P28223 2/20 0.55
DRD3 P35462 2/20 0.55
TMEM97 Q5BJF2 2/20 0.55
SIGMAR1 Q99720 2/20 0.55
ITGB3 P05106 1/20 0.47
ITGA2B P08514 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12403566 0.89 DRD2 (0.68) HRH3HRH1HRH2HTR1ADRD2
SCHEMBL18590696 0.77 CHKA (0.67) HRH3HRH1HRH2SIGMAR1
SCHEMBL7947342 0.77 HRH3 (0.68) HRH3HRH1HRH2ITGB3ITGA2B
SCHEMBL12261943 0.76 DRD4 (0.77) HRH3HRH1DRD2HTR2ADRD3
SCHEMBL12486958 0.74 LTA4H (0.58) HRH3HRH1
SCHEMBL2300940 0.74 LTA4H (0.53) HRH3HRH1
SCHEMBL8696504 0.74 HRH3 (0.51) HRH3HRH1HRH2ITGB3ITGA2B
SCHEMBL8634890 0.73 HRH3 (0.50) HRH3HRH1HRH2ITGB3ITGA2B
SCHEMBL28112415 0.73 CHKA (0.80)
SCHEMBL255055 0.73 ESR1 (0.58) HRH3HTR2ASIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed