SCHEMBL8634628

SCHEMBL8634628

CCOC(=O)Cn1nc(-c2ccc(S(N)(=O)=O)cc2)c(-c2ccc(Cl)cc2Cl)c1C(F)(F)F

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.59
PTGS1 P23219 4/20 0.50
CHRNA7 P36544 4/20 0.45
TSHR P16473 2/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPK1 P28482 1/20 0.43
TRPM2 O94759 1/20 0.43
CNR1 P21554 1/20 0.42
CA9 Q16790 4/20 0.41
CA12 O43570 3/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA4 P22748 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8632536 0.92 PTGS2 (0.70) PTGS2PTGS1TSHRALDH1A1MAPK1
SCHEMBL8631631 0.89 PTGS2 (0.70) PTGS2PTGS1CHRNA7TSHRALDH1A1
SCHEMBL7777880 0.88 PTGS2 (0.50) PTGS2PTGS1CHRNA7CA9CA12
SCHEMBL7777892 0.86 PTGS2 (0.66) PTGS2PTGS1CHRNA7CA9CA12
SCHEMBL8632389 0.84 PTGS2 (0.63) PTGS2PTGS1CHRNA7TRPM2CA9
SCHEMBL8634891 0.84 PTGS2 (0.73) PTGS2PTGS1TSHRALDH1A1TRPM2
SCHEMBL8633238 0.83 PTGS2 (0.84) PTGS2PTGS1CHRNA7TRPM2CA9
SCHEMBL8629917 0.83 PTGS2 (0.72) PTGS2PTGS1TSHRALDH1A1TRPM2
SCHEMBL8634624 0.82 PTGS2 (0.46) PTGS2PTGS1CHRNA7CNR1CA9
SCHEMBL8631062 0.82 PTGS2 (0.67) PTGS2PTGS1CHRNA7TRPM2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed