SCHEMBL8634839

SCHEMBL8634839

C#Cc1ccc2c(c1)NCCC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.40
MAPT P10636 3/20 0.39
KDM4E B2RXH2 2/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
PPARG P37231 3/20 0.36
PPARD Q03181 3/20 0.36
PPARA Q07869 3/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
GAA P10253 1/20 0.36
THRB P10828 1/20 0.36
ALOX15 P16050 1/20 0.36
CASP1 P29466 1/20 0.36
HTT P42858 1/20 0.36
CASP7 P55210 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26923113 0.89 DRD2 (0.40) MAPTALDH1A1GFERTYMS
SCHEMBL8559068 0.86 MAPT (0.50) HRH3MAPTKDM4ECA12CA1
SCHEMBL30480861 0.84 PNMT (0.47) HRH3MAPTKDM4ECA12CA1
SCHEMBL17785608 0.84 PNMT (0.47) HRH3MAPTKDM4ECA12CA1
SCHEMBL23157401 0.74 DRD2 (0.53) HRH3MAPTKDM4ECA12CA1
SCHEMBL8669783 0.72 TSHR (0.40) MAPTCA12CA1CA2ALDH1A1
SCHEMBL9432052 0.72 ALDH1A1 (0.41) CA12CA1CA2ALDH1A1TYMS
SCHEMBL748146 0.72 PNMT (0.55) GFER
SCHEMBL15320816 0.72 MAPT (0.46) HRH3MAPTKDM4ECA12CA1
SCHEMBL596333 0.72 PNMT (0.48) HRH3MAPTKDM4ECA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118259012-A Method for global analysis of functional histidines in proteins 深圳湾实验室 2024-06-28 CN disclosed
CN-104945389-A Xanthone cross-color ketone compound as well as preparation method and application thereof SHANGHAI INST MATERIA MEDICA 2015-09-30 CN disclosed
EP-0825986-A1 QUINOLYL-ETHYNYL DERIVATIVES HAVING RETINOID-LIKE ACTIVITY Allergan (US) 1998-03-04 EP disclosed
US-5616712-A SKIN DISORDERS; ANTICARCINOGENIC AND -INFLAMMATORY AGENTS; AUTOIMMUNE DISEASES; ALLERGAN (US) 1997-04-01 US disclosed
WO-1996036609-A1 QUINOLYL-ETHYNYL DERIVATIVES HAVING RETINOID-LIKE ACTIVITY ALLERGAN (US) 1996-11-21 WO disclosed