SCHEMBL8634928

SCHEMBL8634928

CCCC(=O)C(N)(CN1CCN(c2ccncc2)CC1)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 6/20 0.41
DRD4 P21917 1/20 0.40
SLC6A4 P31645 1/20 0.40
DHFR P00374 1/20 0.39
ITGB3 P05106 3/20 0.39
ITGA2B P08514 3/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
ACHE P22303 1/20 0.38
GRIN2B Q13224 1/20 0.38
P2RX7 Q99572 1/20 0.38
SPHK1 Q9NYA1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634882 0.93 HRH3 (0.42) HRH3DRD4SLC6A4DHFRITGB3
SCHEMBL8634920 0.76 ITGB3 (0.39) HRH3DHFRITGB3ITGA2BCYP2C9
SCHEMBL6600563 0.71 MAPT (0.62) ITGB3ITGA2BCYP3A4CYP2D6CYP2C9
SCHEMBL16546681 0.70 CHKA (0.52) HRH3DHFR
SCHEMBL8699939 0.70 HRH3 (0.44) HRH3DRD4SLC6A4CYP2C9
SCHEMBL8634875 0.70 SPHK1 (0.39) HRH3DRD4SLC6A4ITGB3ITGA2B
SCHEMBL8837987 0.69 ITGB3 (0.63) HRH3DRD4SLC6A4ITGB3ITGA2B
SCHEMBL6180151 0.69 ITGB3 (0.61) HRH3DRD4SLC6A4ITGB3ITGA2B
Hydrochloric Acid SCHEMBL8838017 0.68 ADRB2 (0.39) HRH3ITGB3ITGA2BCYP3A4CYP2D6
SCHEMBL4712908 0.68 CHRNA7 (0.66) HRH3DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed