SCHEMBL8634920

SCHEMBL8634920

CCCC(=O)C(CN)(C(=O)O)N1CCN(c2ccncc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 6/20 0.39
ITGA2B P08514 6/20 0.39
SLC2A1 P11166 3/20 0.38
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
MAPT P10636 2/20 0.37
DHFR P00374 1/20 0.37
TRPV1 Q8NER1 1/20 0.37
HRH3 Q9Y5N1 2/20 0.36
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SPHK1 Q9NYA1 1/20 0.36
USP2 O75604 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634875 0.93 SPHK1 (0.39) ITGB3ITGA2BSLC2A1HRH3SPHK1
SCHEMBL8634928 0.76 HRH3 (0.41) ITGB3ITGA2BCYP2C9DHFRHRH3
Hydrochloric Acid SCHEMBL8838017 0.73 ADRB2 (0.39) ITGB3ITGA2BCYP2C9TSHRHRH3
SCHEMBL8699932 0.72 GAA (0.42) ITGB3ITGA2BCYP2C9TSHRMAPT
SCHEMBL8838135 0.71 ADRB2 (0.40) ITGB3ITGA2BCYP2C9TSHRHRH3
SCHEMBL6600563 0.71 MAPT (0.62) ITGB3ITGA2BCYP2C9TSHRMAPT
SCHEMBL8634882 0.70 HRH3 (0.42) ITGB3ITGA2BDHFRHRH3SPHK1
SCHEMBL8701123 0.68 ADRB2 (0.42) ITGB3ITGA2BCYP2C9TSHRMAPT
SCHEMBL8635008 0.68 ITGB3 (0.44) ITGB3ITGA2BCYP2C9TSHRHRH3
SCHEMBL8837928 0.68 ADRB2 (0.39) ITGB3ITGA2BHRH3SPHK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed