SCHEMBL8635260

SCHEMBL8635260

CCOP(=O)(CC)COc1ccc(CC(C)=O)cc1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.38
KDM4E B2RXH2 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
PDE4A P27815 1/20 0.38
HIF1A Q16665 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
PTPN1 P18031 1/20 0.37
ALOX5 P09917 3/20 0.37
MAPT P10636 3/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
ALDH1A1 P00352 2/20 0.36
LMNA P02545 2/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8758984 0.85 POLB (0.47) POLBSMN1; SMN2KDM4ECYP1A2CYP2D6
SCHEMBL8758970 0.84 POLB (0.46) POLBSMN1; SMN2KDM4ECYP1A2CYP2D6
SCHEMBL9063248 0.79 PTPN1 (0.58) POLBSMN1; SMN2KDM4ECYP1A2CYP2D6
SCHEMBL27833941 0.79 CYP3A4 (0.41) POLBKDM4ENPC1ALDH1A1
SCHEMBL2628188 0.78 POLB (0.59) POLBSMN1; SMN2KDM4ECYP1A2MAPT
SCHEMBL8759406 0.76 KDM4E (0.50) POLBSMN1; SMN2KDM4ECYP1A2CYP2D6
SCHEMBL8634781 0.76 SLC6A4 (0.47)
SCHEMBL8634785 0.76 SLC6A4 (0.47)
SCHEMBL8634784 0.76 SLC6A4 (0.47)
SCHEMBL8635512 0.75 ALDH1A1 (0.46) SMN1; SMN2KDM4EMAPTRAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0717746-B1 PHOSPHINIC ACID DERIVATIVES WITH ANTI-HYPER GLYCEMIC AND/OR ANTI-OBESITY ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1998-07-15 EP disclosed
EP-0717746-A1 PHOSPHINIC ACID DERIVATIVES WITH ANTI-HYPER GLYCEMIC AND/OR ANTI-OBESITY ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1996-06-26 EP disclosed
WO-1995007284-A1 PHOSPHINIC ACID DERIVATIVES WITH ANTI-HYPER GLYCEMIC AND/OR ANTI-OBESITY ACTIVITY SMITHKLINE BEECHAM PLC (GB) 1995-03-16 WO disclosed