SCHEMBL8635293

SCHEMBL8635293

CCCCc1nc(OC)c(OCCOC)n1C(C)(c1ccc(C(C(=O)O)C2CCCC2)cc1)C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 1/20 0.35
ALOX5 P09917 2/20 0.33
HDAC6 Q9UBN7 1/20 0.33
C3AR1 Q16581 1/20 0.32
MMP2 P08253 1/20 0.32
MMP3 P08254 1/20 0.32
MMP9 P14780 1/20 0.32
MMP8 P22894 1/20 0.32
MMP13 P45452 1/20 0.32
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
PTGS2 P35354 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8632769 0.82 CHRM3 (0.35) CHRM3ALOX5HDAC6MMP2MMP3
SCHEMBL8635292 0.69 CHRM3 (0.34) CHRM3ALOX5HDAC6MMP2MMP3
SCHEMBL8632766 0.69
SCHEMBL9010363 0.69
SCHEMBL9010413 0.66
SCHEMBL7835851 0.65 AGTR1 (0.43)
SCHEMBL7839692 0.65 AGTR2 (0.50)
SCHEMBL9010364 0.65 MDM2 (0.35)
SCHEMBL9010387 0.65 CHRM3 (0.35) CHRM3ALOX5HDAC6PTGS2
SCHEMBL8632524 0.64 AGTR1 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776964-A HYPOTENSIVE AGENTS; ANTICHOLESTEROL AGENTS; CARDIOVASCULAR DISORDERS BAYER AKTIENGESELLSCHAFT (DE) 1998-07-07 US disclosed