SCHEMBL8635604

SCHEMBL8635604

O=C(c1ccccc1)c1ccccc1C(=O)N1CSCC1CO

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
AKR1C3 P42330 3/20 0.41
ALDH1A1 P00352 4/20 0.38
HCRTR1 O43613 2/20 0.37
HCRTR2 O43614 2/20 0.37
MAPT P10636 1/20 0.36
PKM P14618 2/20 0.35
ATM Q13315 2/20 0.35
CDC25B P30305 1/20 0.35
HSP90AA1 P07900 1/20 0.35
CCR6 P51684 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TLR9 Q9NR96 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
DRD2 P14416 1/20 0.34
DRD1 P21728 1/20 0.34
DRD3 P35462 1/20 0.34
NR4A1 P22736 1/20 0.34
CYP2C8 P10632 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8638521 0.82 GAA (0.44) GAASMN1; SMN2AKR1C3ALDH1A1MAPT
SCHEMBL8633138 0.79 PREP (0.53) GAAALDH1A1
SCHEMBL8633642 0.77 HCRTR1 (0.53) GAASMN1; SMN2HCRTR1HCRTR2
SCHEMBL8633638 0.77 HCRTR1 (0.53) GAASMN1; SMN2HCRTR1HCRTR2
SCHEMBL23884759 0.68 HSD17B10 (0.41) SMN1; SMN2ALDH1A1HCRTR1HCRTR2NPSR1
SCHEMBL700595 0.67 AKR1C3 (0.85) GAAAKR1C3ALDH1A1MAPTPKM
SCHEMBL29447165 0.67 AKR1C3 (0.85) GAAAKR1C3ALDH1A1MAPTPKM
SCHEMBL3318857 0.67 HCRTR1 (0.40) ALDH1A1HCRTR1HCRTR2
SCHEMBL23884841 0.67 ALDH1A1 (0.37) SMN1; SMN2ALDH1A1HCRTR1HCRTR2
SCHEMBL23884840 0.67 ALDH1A1 (0.37) SMN1; SMN2ALDH1A1HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5847155-A Aromatic pyrrolidine amide prolyl endopeptidase inhibitors PFIZER INC (US) 1998-12-08 US disclosed
EP-0536163-A1 AROMATIC PYRROLIDINE AND THIAZOLIDINE AMIDES PFIZER INC. (US) 1993-04-14 EP disclosed
WO-1991018891-A1 AROMATIC PYRROLIDINE AND THIAZOLIDINE AMIDES PFIZER INC. (US) 1991-12-12 WO disclosed