SCHEMBL8636087

SCHEMBL8636087

CN(C)CCNC(=O)c1cc([N+](=O)[O-])c(N(CCCl)CCCl)c([N+](=O)[O-])c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
GSTP1 P09211 1/20 0.44
GSTM2 P28161 1/20 0.44
ALDH1A1 P00352 7/20 0.42
HPGD P15428 2/20 0.42
HSP90AA1 P07900 1/20 0.42
USP2 O75604 1/20 0.41
PRMT5 O14744 1/20 0.41
WDR77 Q9BQA1 1/20 0.41
HTT P42858 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
POLB P06746 1/20 0.41
LMNA P02545 4/20 0.40
GAA P10253 2/20 0.40
KDM4E B2RXH2 1/20 0.40
GLA P06280 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dimethylamine SCHEMBL8762028 0.85 CYP3A4 (0.42) MAPTSMN1; SMN2ALDH1A1HPGDHSP90AA1
SCHEMBL8636262 0.85 KMT2A (0.46) MAPTSMN1; SMN2GSTP1GSTM2ALDH1A1
SCHEMBL8762462 0.80 ALDH1A1 (0.40) MAPTSMN1; SMN2ALDH1A1HPGDHTT
SCHEMBL8639690 0.79 SMN1; SMN2 (0.43) MAPTSMN1; SMN2GSTP1GSTM2ALDH1A1
SCHEMBL20982472 0.78 SMN1; SMN2 (0.65) MAPTSMN1; SMN2GSTP1GSTM2ALDH1A1
SCHEMBL7474447 0.78 SMN1; SMN2 (0.44) MAPTSMN1; SMN2GSTP1GSTM2ALDH1A1
SCHEMBL2336351 0.78 ALDH1A1 (0.68) MAPTSMN1; SMN2ALDH1A1HPGDHSP90AA1
SCHEMBL8633720 0.76 PARP1 (0.45) MAPTSMN1; SMN2ALDH1A1HTTPOLB
SCHEMBL8635142 0.74 GSTP1 (0.43) MAPTSMN1; SMN2GSTP1GSTM2ALDH1A1
SCHEMBL3583472 0.74 KMT2A (0.44) MAPTSMN1; SMN2ALDH1A1HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750782-A ANTICARCINOGENIC AGENTS, ANTIHYPOXIC AGENTS, PRODRUGS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1998-05-12 US disclosed
EP-0616609-B1 NITROANILINE DERIVATIVES AND THEIR USE AS ANTITUMOR AGENTS CANCER RES CAMPAIGN TECH (GB) 1997-06-18 EP disclosed
US-5571845-A Nitroaniline derivatives and their use as anti-tumour agents CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1996-11-05 US disclosed
EP-0616609-A1 NITROANILINE DERIVATIVES AND THEIR USE AS ANTITUMOR AGENTS. CANCER RES CAMPAIGN TECH (GB) 1994-09-28 EP disclosed
WO-1993011099-A1 NITROANILINE DERIVATIVES AND THEIR USE AS ANTITUMOR AGENTS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1993-06-10 WO disclosed