SCHEMBL8636783

SCHEMBL8636783

CC1(CO)CCCc2ccc(O[Si](c3ccccc3)(c3ccccc3)C(C)(C)C)cc21

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.39
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
CYP3A4 P08684 1/20 0.35
KDM5A P29375 1/20 0.34
KDM4C Q9H3R0 1/20 0.34
KDM5B Q9UGL1 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NR3C1 P04150 4/20 0.32
KDM1A O60341 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8620702 0.93 CYP2C9 (0.34) SIGMAR1CYP2C9TSHRCYP2C19CYP3A4
SCHEMBL8644237 0.92 KDM1A (0.36) SIGMAR1CYP2C19KDM5AKDM4CKDM5B
SCHEMBL8642508 0.82 SIGMAR1 (0.36) SIGMAR1CYP2C9TSHRCYP2C19CYP3A4
SCHEMBL8642502 0.82 SIGMAR1 (0.36) SIGMAR1CYP2C9TSHRCYP2C19CYP3A4
SCHEMBL8586713 0.77 SIGMAR1 (0.31) SIGMAR1
SCHEMBL8586706 0.77 SIGMAR1 (0.31) SIGMAR1
SCHEMBL8641584 0.77 KDM1A (0.34) SIGMAR1KDM1A
SCHEMBL8636777 0.75 SIGMAR1 (0.35) SIGMAR1CYP2C9TSHRCYP2C19CYP3A4
SCHEMBL8615164 0.74 BACE1 (0.32) SIGMAR1
SCHEMBL8612915 0.73 ABL1 (0.34) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998052913-A2 LEUKOTRIENE B4 ANTAGONISTS, IN PARTICULAR 3-OXA-TETRAHYDRONAPHTHALENE-LTB4 ANTAGONISTS SCHERING AKTIENGESELLSCHAFT (DE) 1998-11-26 WO disclosed