SCHEMBL8636972

SCHEMBL8636972

CC(=O)C(CCCS(N)(=O)=O)(c1ccccc1)N1CCN(c2ccncc2)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
HRH3 Q9Y5N1 5/20 0.37
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
LSS P48449 1/20 0.35
SNCA P37840 1/20 0.35
CYP2C9 P11712 2/20 0.35
TSHR P16473 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HIF1A Q16665 1/20 0.35
ITGB3 P05106 1/20 0.35
ITGA2B P08514 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634078 0.82 HRH3 (0.36) CA12CA1CA2CA9HRH3
SCHEMBL8630659 0.76 HTR1A (0.40) HRH3MAPTCYP2C9TSHRCYP2D6
SCHEMBL8702212 0.74 CA12 (0.38) CA12CA1CA2CA9HRH3
SCHEMBL8633904 0.74 ADRB2 (0.36) HRH3CYP2C9TSHRITGB3ITGA2B
SCHEMBL8634084 0.73 CA12 (0.40) CA12CA1CA2CA9HRH3
SCHEMBL8633964 0.72 KDM4E (0.45) HRH3KDM4EGAAMAPTCYP2C9
Hydrochloric Acid SCHEMBL8838192 0.71 KDM4E (0.44) HRH3KDM4EGAAMAPTCYP2C9
SCHEMBL8637197 0.70 MAPT (0.43) HRH3KDM4EGAAMAPTCYP2C9
SCHEMBL8636975 0.69 ITGB3 (0.39) CA12CA1CA2CA9KDM4E
SCHEMBL8686318 0.69 ITGB3 (0.43) CA12CA1CA2CA9HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed