SCHEMBL8637523

SCHEMBL8637523

COc1c(C(=O)c2ccccc2O)ccc(C(=O)N(C)c2ccccc2OCCCCC(=C=O)N2CCN(C)CC2)c1N

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GPR6 P46095 1/20 0.34
RAB9A P51151 1/20 0.32
PTPN1 P18031 1/20 0.31
AVPR2 P30518 1/20 0.31
AVPR1A P37288 1/20 0.31
CDK1 P06493 1/20 0.31
CNR2 P34972 1/20 0.31
DRD3 P35462 1/20 0.31
ALDH1A1 P00352 2/20 0.30
KDM4E B2RXH2 1/20 0.30
POLB P06746 1/20 0.30
MEN1 O00255 1/20 0.30
RAD52 P43351 1/20 0.30
KMT2A Q03164 1/20 0.30
CBX7 O95931 1/20 0.30
HTR1A P08908 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8637529 0.90 AVPR2 (0.40) GPR6RAB9APTPN1AVPR2AVPR1A
SCHEMBL7476396 0.81 CBX7 (0.31) CNR2CBX7
Hydrochloric Acid SCHEMBL7592049 0.80 CBX7 (0.32) ALDH1A1CBX7
SCHEMBL7778674 0.79 KMT2A (0.42) RAB9AAVPR2AVPR1AALDH1A1KDM4E
SCHEMBL7598082 0.79 HRH4 (0.35) DRD3
SCHEMBL7341409 0.78 DRD2 (0.33) GPR6RAB9AAVPR2AVPR1ADRD3
SCHEMBL7781332 0.77 KMT2A (0.39) RAB9AAVPR2AVPR1AALDH1A1KDM4E
SCHEMBL7340721 0.76 AVPR2 (0.39) RAB9AAVPR2AVPR1ACDK1ALDH1A1
SCHEMBL7476543 0.75
SCHEMBL7478475 0.74 CBX7 (0.38) RAB9AAVPR2AVPR1AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832061-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-04-01 EP disclosed