SCHEMBL8638258

SCHEMBL8638258

c1ccc(Cc2ccc(OCCc3ncc[nH]3)cc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.61
LTA4H P09960 11/20 0.60
CYP2D6 P10635 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
HTT P42858 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.47
KMT2A Q03164 1/20 0.46
TSHR P16473 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
LMNA P02545 2/20 0.44
GLA P06280 1/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8641804 0.93 TAAR1 (0.59) TAAR1LTA4HCYP2D6CYP1A2CYP2C9
SCHEMBL8637323 0.88 TAAR1 (0.53) TAAR1LTA4HCYP2D6CYP1A2CYP2C19
SCHEMBL11581355 0.88 TAAR1 (0.53) TAAR1LTA4HCYP2D6CYP1A2CYP2C9
SCHEMBL8639331 0.85 LTA4H (0.49) TAAR1LTA4HCYP2D6CYP1A2CYP2C9
SCHEMBL8685448 0.82 CYP1A2 (0.48) TAAR1LTA4HCYP2D6CYP1A2CYP2C9
SCHEMBL8690542 0.81 CYP3A4 (0.50) TAAR1LTA4HCYP2D6CYP1A2CYP2C9
SCHEMBL11702882 0.81 TAAR1 (0.73) TAAR1LTA4HCYP2D6CYP1A2CYP2C19
SCHEMBL8685427 0.79 GAA (0.56) LTA4HHTTL3MBTL1LMNASMN1; SMN2
SCHEMBL8690250 0.78 HRH3 (0.48) CYP2D6CYP1A2CYP2C9CYP2C19HTT
SCHEMBL8684972 0.78 FPR2 (0.43) TAAR1CYP2D6CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5723492-A LTA4 hydrolase inhibitor pharmaceutical compositions and methods of use G.D. SEARLE & CO. (US) 1998-03-03 US disclosed
US-5719306-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1998-02-17 US disclosed