SCHEMBL8639331

SCHEMBL8639331

c1ccc(Oc2ccc(OCCc3ncc[nH]3)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 7/20 0.49
PLA2G2A P14555 1/20 0.49
TAAR1 Q96RJ0 3/20 0.47
KCNA3 P22001 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP19A1 P11511 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11581355 0.94 TAAR1 (0.53) LTA4HTAAR1KCNA3HRH3CYP1A2
SCHEMBL8637455 0.92 LTA4H (0.51) LTA4HPLA2G2ATAAR1KCNA3HRH3
SCHEMBL8535825 0.90 LTA4H (0.50) LTA4HPLA2G2ATAAR1KCNA3HRH3
SCHEMBL8635977 0.88 LTA4H (0.44) LTA4HCYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL8638258 0.85 TAAR1 (0.61) LTA4HTAAR1CYP1A2CYP2D6CYP2C9
SCHEMBL8637323 0.85 TAAR1 (0.53) LTA4HTAAR1CYP1A2CYP2D6CYP2C19
SCHEMBL8685427 0.81 GAA (0.56) LTA4HHRH3
SCHEMBL8690250 0.81 HRH3 (0.48) HRH3CYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL6181232 0.81 NPC1 (0.49) TAAR1CYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL8684972 0.81 FPR2 (0.43) TAAR1CYP1A2CYP3A4CYP2D6CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5723492-A LTA4 hydrolase inhibitor pharmaceutical compositions and methods of use G.D. SEARLE & CO. (US) 1998-03-03 US disclosed
US-5719306-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1998-02-17 US disclosed